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protein kinase C type-A
Interactions
molecular events
General
PEST protein
protein kinase C (PKC)
Properties
QUALITIES: CATALYTIC-FRAGMENT
SIZE: MW = 78 kD
COMPARTMENT: cytoplasm
STATE: active state
MOTIF: cysteine-rich region
Zinc finger
NAME: Zinc finger (2)
EFFECTOR-BOUND: Zn+2
binding site
EFFECTOR-BOUND: diacylglycerol
C2 domain
MOTIF: allosteric site
EFFECTOR-BOUND: phosphatidylserine
PEST region
EFFECTOR-BOUND: Ca+2
kinase domain
MOTIF: ATP-binding site
NAME: ATP-binding site
MISC-INFO: RECOGNITION-MOTIF
:SEQUENCE XRXX[S*]XRX
:REF " - Kemp BE, Pearson RB.
Protein kinase recognition sequence motifs.
Trends Biochem Sci. 1990 Sep;15(9):342-6. Review.
PMID: 2238044"
INHIBITOR = SPHINGOSINE
References
- Wang KK et al
Calmodulin-binding proteins as calpain substrates.
Biochem J 262:693 1989
PMID: 2556106