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solute carrier family 21 member 14; solute carrier organic anion transporter family member 1C1; organic anion transporter F; OATP-F; organic anion transporter polypeptide-related protein 5; OAT-RP-5; OATPRP5; organic anion-transporting polypeptide 14; OATP-14 (SLCO1C1, OATP14, OATPF, SLC21A14)

Function: - mediates Na+-independent high affinity transport of organic anions such as the thyroid hormones a) thyroxine (T4) b) reverse T3 (rT3) - other potential substrates are transported with much lower efficiency a) triiodothyronine (T3) b) 17-beta-glucuronosyl estradiol c) estrone-3-sulfate d) sulfobromophthalein (BSP) Structure: - belongs to the organo anion transporter (TC 2.A.60) family - contains 1 Kazal-like domain Compartment: membrane Expression: - highly expressed in brain & in Leydig cells in testis - detected in many brain regions - not detected in pons or cerebellum

General

glycoprotein organic anion transporting polypeptide (OATP) solute carrier family 21 (SLC21, SLC21A) transmembrane 10 protein

Properties

SIZE: entity length = 712 aa MW = 79 kD COMPARTMENT: cellular membrane MOTIF: transmembrane domain {80-100} transmembrane domain {111-131} N-glycosylation site {N146} transmembrane domain {222-242} transmembrane domain {270-290} N-glycosylation site {N309} transmembrane domain {353-373} transmembrane domain {393-413} transmembrane domain {427-447} Kazal-type serine protease inhibitor domain {470-525} MOTIF: cysteine residue {X+0} MODIFICATION: cysteine residue {X+X4} cysteine residue {X+X1} MODIFICATION: cysteine residue {X+X3} cysteine residue {X+X2} MODIFICATION: cysteine residue {X+X5} cysteine residue {X+X3} MODIFICATION: cysteine residue {X+X1} cysteine residue {X+X4} MODIFICATION: cysteine residue {X+0} cysteine residue {X+X5} MODIFICATION: cysteine residue {X+X2} N-glycosylation site {N510} N-glycosylation site {N520} FOR-BINDING-OF: serine protease N-glycosylation site {N533} transmembrane domain {550-570} transmembrane domain {592-612} transmembrane domain {643-663} N-glycosylation site {N692}

Database Correlations

OMIM 613389 UniProt Q9NYB5 PFAM correlations Entrez Gene 53919 Kegg hsa:53919

References

UniProt :accession Q9NYB5