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probenecid/sulopenem etzadroxil

Indications: - sulopenem etzadroxil in combination with probenecid to treat uncomplicated urinary tract infections due to certain bacteria in women with limited or no alternative oral antibacterial Contraindications: - blood dyscrasias - uric acid kidney stones Dosage: oral twice daily for 5 days Antimicrobial activity: - Escherichia coli - Klebsiella pneumoniae - Proteus mirabilis Adverse effects: - diarrhea, nausea/vomiting, vulvovaginal yease infection, headache - Clostridioides difficile colitis Drug interactions: - ketorolac tromethamine

General

pharmacologic combination

References

  1. George J FDA Approves Novel Treatment for UTIs New oral antibiotic gets a nod for uncomplicated urinary tract infections. MedPage Today October 25, 2024 https://www.medpagetoday.com/infectiousdisease/generalinfectiousdisease/112596

Components

probenecid (Benemid, Probalan) sulopenem etzadroxil