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FK506-binding protein 1A (12 kD FK506-binding protein, immunophilin FKBP12, FKBP1A)

Function: - may play a role in modulation of ryanodine receptor isoform-1 (RYR-1), a component of the Ca+2 release channel of skeletal muscle sarcoplasmic reticulum - there are 4 molecules of FKBP12 per skeletal muscle RYR. - PPIases accelerate the folding of proteins - catalyzes the cis-trans isomerization of proline imidic peptide bonds in oligopeptides - inhibited by both FK506 & rapamycin peptidylproline (omega=180) peptidylproline (omega=0) Structure: - belongs to the FKBP-type PPIase family, FKBP1 subfamily - contains 1 PPIase FKBP-type domain Compartment: cytoplasm

Interactions

molecular events

Related

FKBP12-rapamycin complex-associated protein; FK506-binding protein 12-rapamycin complex-associated protein 1; rapamycin target protein; RAPT1; mammalian target of rapamycin; mTOR (FRAP1, FRAP, FRAP2)

General

FK506 binding protein (FKBP)

Properties

SIZE: MW = 12 kD entity length = 107 aa COMPARTMENT: cytoplasm MOTIF: active site binding site FOR-BINDING-OF: sirolimus

Database Correlations

OMIM 186945 UniProt P62942 Pfam PF00254 ENZYME 5.2.1.8

References

  1. Martinus RD et al Role of chaperones in the biogenesis and maintenance of the mitochondrion. FASEB J. 1995 Mar;9(5):371-8. Review. PMID: 7896006
  2. UniProt :accession P62942