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norethindrone (Norlutate, Aygestin, Micronor)

Tradenames: Norlutate, Aygestin, Micronor Progestin. Indications: - amenorrhea or abnormal uterine bleeding due to hormonal imbalance - endometriosis - oral contraceptive (alone or in combination with estrogens) Dosage: 5-10 mg PO QD PRN. Tablets: (acetate, Norlutate) 5 mg. Oral Contraceptives: - 0.35 mg QD for 28 days of cycle (28 days) Tablets: (Micronor) 0.35 mg Tablets: (acetate, Norlutate) 5 mg. Adverse effects: 1) common (> 10%) - breakthrough bleeding, spotting, changes in menstrual flow, amenorrhea, pain at site of injection, anorexia, edema, weakness 2) less common (1-10%) - edema, depression, fever, melasma, chloasma, allergic rash with or without pruritus, cholestatic jaundice,changes in cervical erosion & secretions, weight gain or loss, insomnia, breast tenderness

General

progestational agent

Properties

MISC-INFO: elimination route LIVER pregnancy-category D X safety in lactation ?

Database Correlations

PUBCHEM correlations

References

  1. The Pharmacological Basis of Therapeutics, 9th ed. Gilman et al, eds. Permagon Press/McGraw Hill, 1996
  2. Drug Information & Medication Formulary, Veterans Affairs, Central California Health Care System, 1st ed., Ravnan et al eds, 1998
  3. Kaiser Permanente Northern California Regional Drug Formulary, 1998

Component-of

Activella Combipatch estradiol/ethinyl estradiol/ferrous fumarate/iron/norethindrone estradiol/ethinyl estradiol/ferrous fumarate/norethindrone estradiol/ethinyl estradiol/norethindrone estradiol/norethindrone estradiol/norethindrone/relugolix ethinyl estradiol/norethindrone (Junel Fe) ethinyl estradiol/norethindrone/ferrous fumarate (Larin Fe) Femhrt (ethinyl estradiol, norethindrone) Femlyv (ethinyl estradiol, norethindrone) leuprolide/norethindrone Loestrin 24 Fe mestranol/norethindrone Ovcon-35