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multifunctional protein ADE2; phosphoribosylaminoimidazole succinocarboxamide synthase; SAICAR synthetase; phosphoribosylaminoimidazole carboxylase (ADE2, AIRC, PAICS, PAIS)

Function: - purine metabolism; IMP biosynthesis via de novo pathway - 5-amino-1-(5-phospho-D-ribosyl)imidazole-4-carboxamide from N(2)-formyl-N1-(5-phospho-D-ribosyl)glycinamide: step 3/5 - purine metabolism; IMP biosynthesis via de novo pathway - 5-amino-1-(5-phospho-D-ribosyl)imidazole-4-carboxamide from N(2)-formyl-N1-(5-phospho-D-ribosyl)glycinamide: step 4/5 ATP + 5-amino-1-(5-phospho-D-ribosyl)imidazole-4-carboxylate + L-aspartate ADP + phosphate + (S)-2-(5-amino-1-(5-phospho-D-ribosyl)imidazole-4-carboxamido) succinate (SAICAR) 5-amino-1-(5-phospho-D-ribosyl)imidazole-4-carboxylate 5-amino-1-(5-phospho-D-ribosyl)imidazole + CO2 Structure: - homooctamer - synthetase family - carboxylase family

Related

aminoimidazole carboxamide ribonucleotide; 5-amino-1-(5-phospho-D-ribosyl)imidazole-4-carboxamide (AICAR) succinylaminoimidazole carboxamide riboside (SAICAR)

General

carboxy-lyase or decarboxylase ligase or synthetase multifunctional enzyme

Properties

SIZE: entity length = 425 aa MW = 47 kD MOTIF: SAICAR synthetase {2-260} acetylation site SITE: N-TERMINUS EFFECTOR-BOUND: acetyl Ser phosphorylation site {S27} arginine residue {R101} serine residue {S107} Ser phosphorylation site {S107} arginine residue {R215} Thr phosphorylation site {T238} Linker {261-266} AIR carboxylase {267-425} MOTIF: histidine residue {H303} serine residue {S332} glycine residue {G334}

Database Correlations

OMIM 172439 UniProt P22234 PFAM correlations Entrez Gene 10606 Kegg hsa:1060 ENZYME correlations

References

UniProt :accession P22234