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medications contraindicated during pregnancy

Medications labeled pregnancy category X - retinoids a) 13-cis retinoic acid (isotretinoin)* b) all-trans retinoic acid c) etretinate (Tegison) d) tazarotene (Tazorac) e) acitretin (Soriatane) - estrogens a) estradiol b) clomiphene (Clomid) c) dienestrol (Cycladiene) - androgens a) testosterone b) methyltestosterone c) danazol (Danocrine) d) fluoxymesterone (Haloestin, Ora-Testryl) e) nandrolone (Durabolin) f) oxandrolone (Oxandrin) g) stanozolol - progestational agents a) progesterone b) medroxyprogesterone actetate (Provera) c) norethindrone (Norlutate) d) megestrol (Megace) e) norgestrel (Ovrette) f) levonorgestrel (Norplant - gonadotropin-releasing hormone agonists a) goserelin (Zoladex) b) leuprolide (Lupron) c) nafarelin (Synarel) - gonadotropin analogs - urofollitropin (FSH-beta) - finasteride (Proscar) - nicotine - fluorescein - ergot alkaloids a) dihydroergotamine b) methysergide (Sansert) - warfarin* - exception is mechanical heart valve [1] - antineoplastic agents a) 5-fluorouracil (Efudex, 5-FU) b) methotrexate (X) c) mechlorethamine (Mustargen, nitrogen mustard) d) mitomycin C (Mutamycin) e) streptozocin (Zanosar) f) thalidomide* g) flutamide - disease-modifying antirheumatic agents - mycophenolate (D) - leflunomide (X) - cyclophosphamide (D) - benzodiazepines a) estazolam (ProSom) b) flurazepam (Dalmane) c) temazepam (Restoril) d) triazolam (Halcion) e) quazepam (Doral) - statins a) fluvastatin (Lescol) b) lovastatin (Mevacor) c) pravastatin (Pravachol) d) simvastatin (Zocor) e) atorvastatin (Lipitor) f) rosuvastatin (Crestor) g) cerivastatin (Baycol) - antivrals a) ribavirin (Virazole) b) podophyllin (Podofin) - prostaglandin analogs a) misoprostol (Cytotec) b) alprostadil (Muse) - amyl nitrite - combinations a) Bellergal-S or Spastrin (belladonna, phenobarbital, ergotamine) b) conjugated estrogens (Premarin) Management: - mandatory pregnancy prevention program for drugs with *

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pregnancy (gestation) pregnancy category

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medication

References

  1. Medical Knowledge Self Assessment Program (MKSAP) 15, 16. 18. American College of Physicians, Philadelphia 2009, 2012, 2018