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G-protein coupled receptor 182; adrenomedullin receptor (GPR182, ADMR)

Function: orphan receptor Structure: belongs to the G-protein coupled receptor 1 family Compartment: cell membrane Expression: - highly expressed in heart, skeletal muscle, immune system, adrenal gland & liver Note: - originally thought to be a receptor for adrenomedullin [2]

General

glycoprotein G-protein coupled receptor; serpentine receptor

Properties

SIZE: entity length = 404 aa MW = 45 kD COMPARTMENT: cellular membrane MOTIF: exoplasmic domain {1-57} MOTIF: N-glycosylation site {N28} N-glycosylation site {N37} transmembrane domain {58-79} cytoplasmic loop {80-90} transmembrane domain {91-113} exoplasmic loop {114-127} MOTIF: cysteine residue {C126} MODIFICATION: cysteine residue {C202} transmembrane domain {128-149} cytoplasmic loop {150-170} transmembrane domain {171-193} exoplasmic loop {194-217} MOTIF: cysteine residue {C202} MODIFICATION: cysteine residue {C126} transmembrane domain {218-239} cytoplasmic loop {240-258} transmembrane domain {259-280} exoplasmic loop {281-299} transmembrane domain {300-320} cytoplasmic domain {321-404}

Database Correlations

OMIM 605307 UniProt O15218 Pfam PF00001 Entrez Gene 11318 Kegg hsa:1131

References

  1. UniProt :accession O15218
  2. Hanze J et al Molecular cloning of a novel human receptor gene with homology to the rat adrenomedullin receptor and high expression in heart and immune system. Biochem Biophys Res Commun. 1997 Nov 7;240(1):183-8 PMID: 9367907