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Specific
1-[5-Isoquinoline-sulfonyl]-2-methylpiperazine-dihydrochloride (H7)
1-[5-Isoquinoline-sulfonyl]-3-methylpiperazine-dihydrochloride (iso H7)
14-3-3 protein beta/alpha; protein kinase C inhibitor protein 1; KCIP-1; protein 1054 (YWHAB)
20S proteasome inhibitor
5,8,11,14-eicosatetraynoic acid
5-alpha reductase inhibitor
abametapir (Xeglyze)
abiraterone acetate (Zytiga)
acetohydroxamic acid (Lithostat)
actinomycin A
AEBSF (Pefabloc SC, 4-[2-aminoethyl]benzenesulfonyl fluoride)
aldose reductase inhibitor
allopurinol (Zyloprim, Lopurin, Zurinol)
alpha glucosidase inhibitor
amanitin
amastatin
amrinone (Inocor, inamrinone)
anthracycline
antineoplastic enzyme inhibitor
antizyme inhibitor 1; AZI; ornithine decarboxylase antizyme inhibitor (AZIN1, OAZI, OAZIN)
aramchol
aromatase inhibitor
arphamenine-A
arrestin
atabecestat
avasimibe
batimastat
bedaquiline (Sirturo)
belinostat (Beleodaq)
bempedoic acid (Nexletol)
benserazide (Serazide)
beta-lactamase inhibitor
bivalirudin (Angiomax)
calcineurin inhibitor
calcipressin
calyculin A
carbidopa (Lodosyn)
carbonic anhydrase inhibitor
Caspase-1 inhibitor INCA; inhibitory caspase recruitment domain protein (INCA, CARD17)
cedazuridine
cholinesterase inhibitor
cilastatin
cilostazol (Pletal)
Clara cell phospholipid-binding protein; uteroglobin; CCPBP; Clara cells 10 kD secretory protein; CC10; secretoglobin family 1A member 1; urinary protein 1; UP-1; UP1; urine protein 1 (SCGB1A1, CC10, CCSP, UGB)
coagulation factor Xa inhibitor
cobimetinib
coumaran; furocoumaran
dabrafenib (Tafinlar)
darapladib
dasabuvir
deleobuvir
diarylquinolone
dirlotapide (Slentrol)
ecallantide (Kalbitor)
elafin; elastase-specific inhibitor; ESI; peptidase inhibitor 3; PI-3; protease inhibitor WAP3; skin-derived antileukoproteinase; SKALP; WAP four-disulfide core domain protein 14 (PI3, WAP3, WFDC14)
entacapone (Comtan)
epipodophyllotoxin
febuxostat (Uloric)
flavopiridol
fluoroquinolone
folate antagonist; folic acid analog; folic acid antagonist
fondaparinux (Arixtra)
fostamatinib (Tavalisse)
GDP dissociation inhibitor (GDI)
givinostat (Duvyzat)
gliptin; dipeptidyl peptidase-4 inhibitor; DPP-4 inhibitor
histone decetylase inhibitor
HMG CoA reductase inhibitor (statin)
hydroxyurea; hydroxycarbamide (Hydrea, Droxia)
hypericin
inhibitor of Bruton tyrosine kinase (IBTK, BTKI, KIAA1417)
inhibitor of metalloproteinase (IMP) or tissue inhibitor of metalloproteinase (TIMP)
inosine-5'-monophosphate dehydrogenase inhibitor; IMP dehydrogenase inhibitor
integrase inhibitor; integrase strand transfer inhibitor (InSTI)
ivosidenib (Tibsovo)
J147
kinase inhibitor
latexin (endogenous carboxypeptidase inhibitor, ECI, tissue carboxypeptidase inhibitor, TCI, MUM, LXN)
leflunomide; teriflunomide (Arava)
lesinurad (Zurampic)
lipocortin or calpactin
lipoxygenase inhibitor
lonafarnib (Sarasar)
ly294002
maralixibat; lopixibat (Livmarli)
mavacamten (Camzyos)
metyrosine (Demser)
miglustat (Acetlion, Zavesca, Opfolda)
milrinone (Primacor Corotrope)
mitoxantrone (Novantrone, Mitozantrone)
monoamine oxidase [MAO] inhibitor
neprilysin inhibitor
neuraminidase inhibitor
non-steroidal anti-inflammatory agent (NSAID)
NS5A inhibitor
odevixibat (Bylvay)
opicapone (ONGENTYS)
orlistat (Xenical, Alli)
ornithine decarboxylase antizyme
paroxon; paraoxon
PARP inhibitor
PCSK9 inhibitor (ALN-PCS)
pegaptanib
pentostatin (Nipent, DCF, 2'deoxycoformycin)
peptidase inhibitor 16 (cysteine-rich secretory protein 9, CRISP-9, PSP94-binding protein, PI16, CRISP9, PSPBP, UNQ289/PRO328)
phenylarsine oxide; oxyphenylarsine
phosphatase inhibitor
phosphodiesterase inhibitor
protease inhibitor
Protein phosphatase inhibitor 2-like protein 1 (protein phosphatase 1 regulatory subunit 2 pseudogene 1, PPP1R2P1)
protein phosphatase inhibitor 2-like protein 3 (protein phosphatase 1 regulatory subunit 2 pseudogene 3, PPP1R2P3)
protein synthesis inhibitor
proteinase inhibitor E-64 (thiol protease inhibitor E-64, Lopac E-3132)
proton pump inhibitor
pyrimidine synthesis inhibitor
ras GTPase inhibitor
retenone
reuptake inhibitor
reverse transcriptase inhibitor (RTI)
ribonuclease inhibitor; ribonuclease/angiogenin inhibitor 1; RAI; placental ribonuclease inhibitor; Rnase inhibitor; RI (RNH1, PRI, RNH)
ruxolitinib (Jakafi, Opzelura)
semagacestat
serotonin-2 antagonist-reuptake inhibitor (SARI)
SGLT-2 inhibitor; oral glucosuric agent; flozin
suicide inhibitor
taselisib
telotristat; telotristat ethyl (Xermelo)
TG101348
thapsigargin
thrombin inhibitor
tipiracil
tolcapone (Tasmar)
topoisomerase inhibitor
trametinib (Mekinist)
tribbles homolog 1 (TRB-1, SKIP1, G-protein-coupled receptor-induced protein 2, GIG-2, TRIB1, C8FW, GIG2, TRB1)
tribbles homolog 2 2 (TRB-2, TRIB2, TRB2)
triclosan (Irgasan, Cloxifenolum, Triclosanum, Cliniclean, Cloxifenol, Tersaseptic, Aquasept, Manusept, Sapoderm)
trilostane (Vetoryl)
vadadustat
vascular endothelial growth factor (VEGF) inhibitor
verubecestat
viral helicase primase inhibitor
wortmannin
zoliflodacin (ETX0914)
General
bioagent