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avacincaptad pegol (Izeray)

Indications: - geographic atrophy secondary to age-related macular degeneration Dosage: - 2 mg, 0.1 mL of 20 mg/mL solution intravitreal injection once monthly - for use up to 12 months 20 mg/mL in single-dose vial Adverse effects: - most common - conjunctival hemorrhage (13%) - increased intraocular pressure (9%) - blurred vision (8%) - neovascular age-related macular degeneration (7%) - other - endophthalmitis - retinal detachment Mechanism of action: - complement inhibitor - PEGylated oligonucleotide that binds to & inhibits complement C5 - by inhibiting C5, avacincaptad pegol may prevent its cleavage to C5a & C5b thus decreasing membrane attack complex (MAC) formation.

General

ophthalmic agent (eyedrops)

References

  1. HIGHLIGHTS OF PRESCRIBING INFORMATION Izeray (avacincaptad pegol intravitreal solution) https://ivericbio.com/wp-content/uploads/IZERVAY-avacincaptad-pegol-intravitreal-solution-PI_Final_8.4.23.pdf