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multidrug resistance-associated protein 6; ATP-binding cassette sub-family C member 6; anthracycline resistance-associated protein; multi-specific organic anion transporter E; MOAT-E (ABCC6 ARA MRP6)

Function: - may participate directly in the active transport of drugs into subcellular organelles or influence drug distribution indirectly - transports glutathione conjugates including leukotriene-C4 (LTC4) & N-ethylmaleimide S-glutathione (NEM-GS) Structure: - belongs to the ABC transporter family, conjugate transporter (TC 3.A.1.208) subfamily - contains 2 ABC transmembrane type-1 domains; residues 311-593 & 947-1228 - contains 2 ABC transporter domains; residues 629-853 & 1265-1499 Compartment: membrane Expression: - expressed in kidney & liver - very low expression in other tissues Pathology: - defects in ABCC6 are the cause of pseudoxanthoma elasticum

General

ATP-binding cassette sub-family C (ABC transporter-C, ABCC) glycoprotein phosphoprotein transmembrane 17 protein

Properties

SIZE: entity length = 1503 aa MW = 165 kD COMPARTMENT: cellular membrane MOTIF: exoplasmic domain {1-31} MOTIF: N-glycosylation site {N15} transmembrane domain {32-52} cytoplasmic loop {53-72} transmembrane domain {73-93} exoplasmic loop {94-98} transmembrane domain {99-119} cytoplasmic loop {120-131} transmembrane domain {132-149} exoplasmic loop {150-167} transmembrane domain {168-188} cytoplasmic loop {189-302} MOTIF: Ser phosphorylation site {S244} transmembrane domain {303-323} exoplasmic loop {324-349} transmembrane domain {350-370} cytoplasmic loop {371-426} transmembrane domain {427-447} exoplasmic loop {448-450} transmembrane domain {451-471} cytoplasmic loop {472-533} transmembrane domain {534-554} exoplasmic loop {555-575} transmembrane domain {576-596} cytoplasmic loop {597-939} MOTIF: ATP-binding site NAME: ATP-binding site SITE: 663-670 Ser phosphorylation site {S902} transmembrane domain {940-960} exoplasmic loop {961-997} transmembrane domain {998-1018} cytoplasmic loop {1019-1061} transmembrane domain {1062-1082} exoplasmic loop {1083-1083} transmembrane domain {1084-1104} cytoplasmic loop {1105-1175} transmembrane domain {1176-1196} exoplasmic loop {1197-1198} transmembrane domain {1199-1219} cytoplasmic domain {1220-1503} MOTIF: ATP-binding site NAME: ATP-binding site SITE: 1299-1306

Database Correlations

OMIM correlations MORBIDMAP 603234 UniProt O95255 PFAM correlations Entrez Gene 368

References

  1. UniProt :accession O95255
  2. Mutations of the ABCC6 gene Retina International's Scientific Newsletter http://www.retina-international.com/sci-news/abcc6mut.htm
  3. GeneReviews https://www.genecards.org/cgi-bin/carddisp.pl?gene=ABCC6