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ubiquitin-activating enzyme E1 (ubiquitin-like modifier-activating enzyme 1, A1S9 protein, UBE1, UBA1, A1S9T)

Function: - catalyzes 1st step of ubiquitin conjugation, ligation of the C-terminal Gly of ubiquitin with Cys within UBE1 (itself), yielding an ubiquitin-E1 thioester & free AMP - protein degradation; protein ubiquitinylation Structure: - monomer (putative) - belongs to the ubiquitin-activating E1 family - there are 2 active sites within the E1 molecule, allowing it to accommodate 2 ubiquitin moieties at a time, with a new ubiquitin forming an adenylate intermediate as the previous one is transferred to the thiol site

Related

NEDD8-activating enzyme E1 catalytic subunit; NEDD8-activating enzyme E1C; ubiquitin-activating enzyme E1C; ubiquitin-like modifier-activating enzyme 3; ubiquitin-activating enzyme 3 (UBA3, UBE1C) ubiquitin-activating enzyme E1 homolog (ubiquitin-like modifier-activating enzyme 7, UBA7, UBE2, UBE1L)

Specific

ubiquitin-like modifier-activating enzyme 5; ubiquitin-activating enzyme 5; thiFP1; UFM1-activating enzyme; ubiquitin-activating enzyme E1 domain-containing protein 1 (UBA5, UBE1DC1)

General

ligase or synthetase phosphoprotein

Properties

SIZE: entity length = 1058 aa MW = 118 kD MOTIF: Ser phosphorylation site {S46} Tyr phosphorylation site {Y55} 2 approximate repeats {63-611} MOTIF: consensus repeat {63-199} consensus repeat {459-611} ATP-binding site NAME: ATP-binding site SITE: 478-507 cysteine residue {C632}

Database Correlations

OMIM 314370 MORBIDMAP 314370 UniProt P22314 PFAM correlations Entrez Gene 7317 Kegg hsa:7317

References

  1. Jentsch et al TIBS 15(May):195 1990
  2. UniProt :accession P22314