Search
tyrosine kinase inhibitor
Monitor:
- periodic ECG monitoring
Adverse effects:
- hypertension, may be severe [1]
- all tyrosine kinase inhibitors can prolong QT interval [1]
Specific
acalabrutinib (Calquence)
antineoplastic tyrosine kinase inhibitor
avapritinib (Ayvakit)
brigatinib (Alunbrig)
capmatinib (Tabrecta)
erbstatin
genistein
gilteritinib (Xospata)
herbimycin A
Janus kinase inhibitor; JAK inhibitor
lavendustin A
midostaurin (Rydapt)
mobocertinib (Exkivity)
oclacitinib maleate (Apoquel)
pemigatinib (Pemazyre)
pralsetinib (Gavreto)
quercetin
selpercatinib (Retevmo)
tyrphostin
General
protein kinase inhibitor
Properties
INHIBITS: protein kinase
References
- Medical Knowledge Self Assessment Program (MKSAP) 17,
American College of Physicians, Philadelphia 2015