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somatostatin receptor
Related
somatostatin; growth hormone release-inhibiting factor; contains: somatostatin-28, somatostatin-14 (SST)
Specific
somatostatin receptor 1; SS1R; SRIF-2 (SSTR1)
somatostatin receptor 2; SS2R; SRIF-1 (SSTR2)
somatostatin receptor 3; SS3R; SSR-28 (SSTR3)
somatostatin receptor 4; SS4R; brain-specific somatostatin receptor (SSTR4)
somatostatin receptor 5; SS5R (SSTR5)
General
G-protein coupled receptor; serpentine receptor
synaptic receptor
Properties
COMPARTMENT: synaptic membrane
CELL: neuron
MOTIF: exoplasmic domain {N-TERMINAL}
transmembrane domain {TM1}
transmembrane domain {TM2}
transmembrane domain {TM3}
transmembrane domain {TM4}
transmembrane domain {TM5}
transmembrane domain {TM6}
transmembrane domain {TM7}
binding site
SITE: C-TERMINAL-CYS
EFFECTOR-BOUND: palmitate
BOUND-VIA: carboxylate
cytoplasmic domain {C-TERMINAL}
References
- VanDongen AM, Codina J, Olate J, Mattera R, Joho R,
Birnbaumer L, Brown AM.
Newly identified brain potassium channels gated by the guanine
nucleotide binding protein Go.
Science. 1988 Dec 9;242(4884):1433-7.
PMID: 3144040
- prosite :accession PS00237