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SKP1-CUL1-F-box protein (SCF) complex; SCF(FBXW11) E3 ligase complex; CF(SKP2) E3 ligase complex

Function: - mediates ubiquitination & subsequent proteasomal degradation of target proteins involved in cell cycle progression, signal transduction & transcription - recognizes phosphorylated CDKN1B/p27kip & is involved in regulation of G1/S transition Structure: - consists of CUL1, RBX1, SKP1, SKP2, FBXL (FBXL19, FBXL21, FBXW9, FBXW12)

Related

E3 ubiquitin ligase; ubiquitin-ligating enzyme E3; N end-recognizing protein

General

SCF-type E3 ligase complex

Properties

SUBUNITS: S-phase kinase-associated protein 1 MOTIF: F-box interaction {104-163} S-phase kinase-associated protein 2 MOTIF: Ser phosphorylation site {S64} F-box domain {94-140} Ser phosphorylation site {S179} leucine-rich repeat SITE: 180-204 MOTIF: leucine residue (SEVERAL) leucine-rich repeat SITE: 210-234 MOTIF: leucine residue (SEVERAL) leucine-rich repeat SITE: 258-284 MOTIF: leucine residue (SEVERAL) leucine-rich repeat SITE: 286-308 MOTIF: leucine residue (SEVERAL) leucine-rich repeat SITE: 309-330 MOTIF: leucine residue (SEVERAL) leucine-rich repeat SITE: 334-356 MOTIF: leucine residue (SEVERAL) leucine-rich repeat SITE: 359-378 MOTIF: leucine residue (SEVERAL) leucine-rich repeat SITE: 380-403 MOTIF: leucine residue (SEVERAL) cullin 1 COMPARTMENT: synaptic membrane CELL: neuron MOTIF: membrane region binding site SITE: 720-720 FOR-BINDING-OF: ubiquitin RING-box protein 1 COMPARTMENT: cytoplasm cell nucleus MOTIF: acetylation site SITE: N-TERMINUS EFFECTOR-BOUND: acetyl Ser phosphorylation site {S11} Zn+2-binding site SITE: 42-42 Zn+2-binding site SITE: 45-45 RING-finger {53-98} MOTIF: Zn+2-binding site SITE: 53-53 Zn+2-binding site SITE: 56-56 Zn+2-binding site SITE: 68-68 Zn+2-binding site SITE: 75-75 Zn+2-binding site SITE: 77-77 Zn+2-binding site SITE: 80-80 Zn+2-binding site SITE: 82-82 Zn+2-binding site SITE: 83-83 Zn+2-binding site SITE: 94-94 Zn+2-binding site SITE: 97-97 EFFECTOR-BOUND: Zn+2 FOR-BINDING-OF: DNA motif F-box & leucine-rich repeat protein MOTIF: F-box domain leucine-rich repeat MOTIF: leucine residue (SEVERAL) cullin-associated NEDD8-dissociated protein 1 COMPARTMENT: cell nucleus MOTIF: HEAT repeat {2-39} acetylation site SITE: N-TERMINUS EFFECTOR-BOUND: acetyl HEAT repeat {44-81} HEAT repeat {83-119} HEAT repeat {131-165} HEAT repeat {171-208} HEAT repeat {210-247} HEAT repeat {248-282} HEAT repeat {289-366} MOTIF: Ser phosphorylation site {S335} Ser phosphorylation site {S340} HEAT repeat {370-407} HEAT repeat {424-467} HEAT repeat {471-510} HEAT repeat {515-552} HEAT repeat {563-602} HEAT repeat {606-643} MOTIF: Thr phosphorylation site {T624} HEAT repeat {646-683} HEAT repeat {688-725} HEAT repeat {729-768} HEAT repeat {770-808} HEAT repeat {809-845} HEAT repeat {852-889} HEAT repeat {890-927} HEAT repeat {928-960} HEAT repeat {961-998} HEAT repeat {1002-1039} HEAT repeat {1043-1097} HEAT repeat {1099-1133} HEAT repeat {1140-1189}

References

  1. UniProt :accession P34991
  2. UniProt :accession Q13309

Components

cullin homolog 1 (CUL-1) cullin-associated NEDD8-dissociated protein 1; cullin-associated & neddylation-dissociated protein 1; TBP-interacting protein of 120 kD A; TBP-interacting protein 120A; p120 CAND1 (CAND1, KIAA0829, TIP120, TIP120A) F-box & leucine-rich repeat protein RING-box protein 1; Rbx1; regulator of cullins 1; RING finger protein 75; protein ZYP (RBX1 RNF75 ROC1) S-phase kinase-associated protein 1; cyclin-A/CDK2-associated protein p19; p19skp1; p19A; RNA polymerase II elongation factor-like protein; organ of corti protein 2; OCP-2; organ of corti protein II; OCP-II; transcription elongation factor B; SIII (SKP1, EMC19, OCP2, SKP1A, TCEB1L) S-phase kinase-associated protein 2; F-box protein Skp2; cyclin-A/CDK2-associated protein p45; p45skp2; F-box/LRR-repeat protein 1 (SKP2 FBXL1)