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rho-associated kinase ROCK

two isoforms: ROCK1 & ROCK2. Function: - downstream effector of Rho proteins - role in cytokeletal assembly & reorganization - both ROCK1 & ROCK2 negativel regulate of VEGF-induced angiogenic endothelial cell activation Comparative biology: - IL-17 facilitates Rho-kinase dependent inhibitory phosphorylation of endothelial nitric oxide synthase in mice reducing nitric oxide production in cerebral endothelial cells, inhibiting resting cerebral perfusion & endothelial function, leading to cognitive impairment* [2] * unclear if this is ROCK1, ROCK2 or both [2]

Specific

rho-associated coiled-coil-containing protein kinase 1; p160ROCK; ROK-beta; Rho-associated protein kinase 1 (ROCK1) Rho-associated protein kinase 2; Rho kinase 2; Rho-associated, coiled-coil-containing protein kinase 2; p164 ROCK-2 (ROCK2, KIAA0619)

General

serine/threonine kinase

Properties

STATE: active state MOTIF: S/T phosphorylation site kinase domain MOTIF: ATP-binding site NAME: ATP-binding site

References

  1. Zhao Z, Rivkees SA. Rho-associated kinases play a role in endocardial cell differentiation and migration. Dev Biol. 2004 Nov 1;275(1):183-91. PMID: 15464581
  2. Faraco G, Brea D, Garcia-Bonilla L. Dietary salt promotes neurovascular and cognitive dysfunction through a gut-initiated TH17 response. Nature Neuroscience. Jan 15, 2018 PMID: 29335605 https://www.nature.com/articles/s41593-017-0059-z