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eletriptan (Relpax)

Pharmacokinetics: 1) may have faster onset than sumatriptan 2) metabolized by cyt P450 3A4 Drug interactions: -> cyt P450 3A4 inhibitors increase eletriptan -> clarithromycin (Biaxin), ketoconazole (Nizoral), itraconazole (Sporonox), nefazodone (Serzone), ritonavir (Norvir), nelfinavir (Viracept)

Interactions

drug interactions drug adverse effects of triptan(s)

General

serotonin agonist (5-HT receptor agonist, triptan)

Database Correlations

PUBCHEM correlations

References

  1. Prescriber's Letter 10(3):14 2003
  2. Pfizer