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eletriptan (Relpax)
Pharmacokinetics:
1) may have faster onset than sumatriptan
2) metabolized by cyt P450 3A4
Drug interactions:
-> cyt P450 3A4 inhibitors increase eletriptan
-> clarithromycin (Biaxin), ketoconazole (Nizoral), itraconazole (Sporonox), nefazodone (Serzone), ritonavir (Norvir), nelfinavir (Viracept)
Interactions
drug interactions
drug adverse effects of triptan(s)
General
serotonin agonist (5-HT receptor agonist, triptan)
Database Correlations
PUBCHEM correlations
References
- Prescriber's Letter 10(3):14 2003
- Pfizer