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Specific
adenosine A2A receptor antagonist
adrenergic receptor antagonist
androgen receptor antagonist; androgen receptor signaling inhibitor (ARSI)
angiotensin II receptor antagonist (ARB)
avacopan
betahistine
brodalumab (Siliq)
cannobinoid receptor antagonist
CCR5 antagonist
cenicriviroc
degarelix (Firmagon)
elinzanetant
endothelin receptor antagonist
etrasimod (Velsipity)
fezolinetant (Veozah)
gamma aminobutyrate (GABA) antagonist
glycoprotein IIb/IIIa inhibitor
icatibant (Firazyr)
IL-6 receptor inhibitor
lemborexant (Dayvigo)
leukotriene receptor antagonist
lymphocyte function-associated antigen 1 (LFA-1) antagonist
nefazodone (Serzone, Dutonin, Nefador, Nefirel, Rezeril)
netupitant; fosnetupitant
NMDA receptor antagonist
opioid receptor antagonist or narcotic antagonist
ozanimod (Zeposia)
P2Y12-receptor inhibitor
perampanel (Fycompa)
revacept
rilonacept (Arcalyst)
serotonin antagonist
StemRegenin 1 (SR1)
strychnine
ticlopidine (Ticlid)
vasopressin receptor antagonist (vaptan)
vorapaxar (Zontivity)
General
bioagent