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phosphodiesterase-4 inhibitor
Indications:
- inhibitors of PDE4 are used for treatment of COPD. Mmechanism of action:
- molecule inhibiting phosphodiesterase-4
Specific
apremilast (Otezla)
crisaborole (Eucrisa)
ensifentrine (Ohtuvayre)
roflumilast (Daliresp)
RPL554
General
bronchodilator
phosphodiesterase inhibitor
Properties
INHIBITS: phosphodiesterase 4
References
- Beghe B, Rabe KF, Fabbri LM.
Phosphodiesterase-4 inhibitor therapy for lung diseases.
Am J Respir Crit Care Med. 2013 Aug 1;188(3):271-8. Review.
PMID: 23656508
- Chong J, Leung B, Poole P.
Phosphodiesterase 4 inhibitors for chronic obstructive pulmonary disease.
Cochrane Database Syst Rev. 2017 Sep 19;9:CD002309. Review.
PMID: 28922692