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Ovral (ethinyl estradiol/norgestrel)

50 ug ethinyl estradiol (estrogen) plus 0.5 mg norgestrel (progestin) Indications: - postcoital contraception (morning after pill) * levonorgestrel 1.5 mg (One Step now advertised on WebMD) & ulipristal are used [3] (see morning after pill) Contraindications: pregnancy-category X safety in lactation - Dosage: 1) 2 tablets at 1st visit 2) 2 tablets 12 hours later Pharmacokinetics: elimination: liver Adverse effects: 1) common (> 10%) - nausea, peripheral edema, breast enlargement, breast tenderness, anorexia, bloating 2) not common (1-10%) - vomiting, diarrhea, increased libido, headache 3) uncommon (< 1%) - intolerance to contact lenses, breast tumors, amenorrhea, alterations in mestrual flow, hypertension, thromboembolism, stroke, myocardial infarction, edema, depression, dizziness, anxiety, chloasma, melasma, rash, hyperglycemia, GI distress, increased serum triglycerides, increased LDL, cholestatic jaundice, increased susceptibility to Candida infection Drug interactions: - barbiturates, carbamazepine, cyclosporine, griseofulvin, penicillins, phenytoin, rifampin, tetracyclines

Interactions

drug adverse effects of estrogens

General

monophasic oral contraceptive ethinyl estradiol/norgestrel

References

  1. Kaiser Permanente Northern California Regional Drug Formulary, 1998
  2. WebMD Plan B One-Step http://www.webmd.com/sex/birth-control/plan-b#1
  3. Locke T for Medscape. Sept 21, 2016 Emergency Contraceptives Affected by Other Medications, UK Warns. http://www.medscape.com/viewarticle/869116