Search
chloroprocaine (Nesacaine)
Tradename: Nesacaine.
Indications:
1) local anesthesia
2) epidural anesthesia
Contraindications:
1) myasthenia gravis
2) concurrent use of bupivicaine
3) NOT for subarachnoid administration
Caution:
1) cardiac disease
2) hypothyroidism
Dosage: 1%, 2%, 3%.
Adverse effects:
- uncommon (< 1%)
- myocardial depression, hypotension, bradycardia, edema, cardiovascular shock, anxiety, restlessness, disorientation, confusion, tremors, shivering, seizures, drowsiness, loss of consciousness, urticaria, nausea/vomiting, transient burning at the injection site, blurred vision, tinnitus, respiratory arrest, anaphylactoid reaction, chills
General
local anesthetic
Properties
MISC-INFO: elimination route LIVER
KIDNEY
Database Correlations
PUBCHEM correlations
References
- The Pharmacological Basis of Therapeutics, 9th ed.
Gilman et al, eds. Permagon Press/McGraw Hill, 1996
- Kaiser Permanente Northern California Regional Drug
Formulary, 1998