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metformin/sitagliptin; januvia/metformin (Janumet)

Indications: - treatment of diabetes mellitus type 2 Contraindications: - renal failure: eGFR < 30 mL/min/1.73 m2 - metabolic acidosis - not for use in treatment of diabetes mellitus type 1 Dosage: - BID dosing - 50 mg sitagliptin + 500 mg or 1000 mg metformin

Interactions

drug adverse effects of hypoglycemic agents

General

hypoglycemic combination

References

  1. Prescriber's Letter 14(5): 2007 Januvia's Place in Therapy Detail-Document#: 230511 (subscription needed) http://www.prescribersletter.com
  2. Highlights of Prescribing Information JanuMet (sitagliptin & metformin extended release) for oral use https://www.merck.com/product/usa/pi_circulars/j/janumet/janumet_pi.pdf - Highlights of Prescribing Information JanuMet XR (sitagliptin & metformin hydrochloride) for oral use https://www.merck.com/product/usa/pi_circulars/j/janumet_xr/janumet_xr_pi.pdf

Components

metformin (Glucophage) sitagliptin (Januvia)