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lemborexant (Dayvigo)
Indications:
- insomnia
Contraindications:
- narcolepsy [2]
Dosage:
- 5-10 mg
Tabs: 5 mg, 10 mg
Pharmacokinetics:
- elimination 1/2life 17-19 hours [2]
Adverse effects:
- next-day somnolence
- impaired driving
- cataplexy-like symptoms [2]
Mechanism of action:
- orexin receptor antagonist
General
sleeping pill
receptor antagonist
Database Correlations
PUBCHEM cid=56944144
References
- Remaly J
FDA Approves Lemborexant (Dayvigo) for Insomnia.
Medscape - Dec 23, 2019.
https://www.medscape.com/viewarticle/923054
- Talebraza S et al
Geriatrics Evaluation & Management Tools
American Geriatrics Society. 2021
https://geriatricscareonline.org/ProductAbstract/geriatrics-evaluation-management-tools/B007/