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dasabuvir/ombitasvir/paritaprevir/ritonavir (Viekira XR)

Indications: - hepatitis C infection genotype 1 Contraindications: - concurrent use of ethinyl estradiol - moderate to severe hepatic impairment (Child-Pugh class B & C) Adverse effects: - fatigue - asthenia - nausea, - insomnia - pruritus & other skin reactions - hepatoxicity [3] - elevated serum transaminases (5-fold elevation in 1%) - reactivation of hepatitis B in patients with current or previous hepatitis B infection [2] - 24% of patients with chronic hepatitis B [3] - 1.4% with resolved hepatitis B infection [3] Drug interactions: - contraceptives containing ethinyl estradiol increase likelihood of increased serum transaminases - proton pump inibitors have no effect on efficacy Notes: - manufacturer: Abbvie

Interactions

drug interactions

Related

ombitasvir/paritaprevir/ritonavir (Viekira, Technivie)

General

antiviral combination

References

  1. FDA Approves Single-Tablet Viekira XR for Hepatitis C. Medscape. Jul 26, 2016. http://www.medscape.com/viewarticle/866680
  2. FDA Drug Safety Communication: Oct 4, 2016 FDA warns about the risk of hepatitis B reactivating in some patients treated with direct-acting antivirals for hepatitis C. http://www.fda.gov/Drugs/DrugSafety/ucm522932.htm
  3. Mucke MM, Backus LI, Mucke VT et al Hepatitis B virus reactivation during direct-acting antiviral therapy for hepatitis C: a systematic review and meta-analysis. Lancet Gastroenterology & Hepatology. Jan 19, 2018 PMID: 29371017 http://www.thelancet.com/journals/langas/article/PIIS2468-1253(18)30002-5/fulltext

Components

dasabuvir ombitasvir paritaprevir ritonavir (Norvir, RTV)