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cannabinoid receptor
Function:
- coupled to Gi
- endogenous ligand is anandamide.
Related
anandamide
Gi-protein
Specific
cannabinoid receptor 1; CB1; CB-R; CANN6 (CNR1, CNR)
cannabinoid receptor 2; CB-2; CB2; CX5 (CNR2)
General
G-protein coupled receptor; serpentine receptor
Properties
COMPARTMENT: cellular membrane
MOTIF: exoplasmic domain {N-TERMINAL}
ligand-binding site
FOR-BINDING-OF: anandamide
transmembrane domain {TM1}
transmembrane domain {TM2}
transmembrane domain {TM3}
transmembrane domain {TM4}
transmembrane domain {TM5}
transmembrane domain {TM6}
transmembrane domain {TM7}
transmembrane domain (7)
guanine nucleotide exchange domain
NAME: guanine nucleotide exchange domain
binding site
SITE: C-TERMINAL-CYS
EFFECTOR-BOUND: palmitate
BOUND-VIA: carboxylate
cytoplasmic domain {C-TERMINAL}
MISC-INFO: LIGAND = ANANDAMIDE
Database Correlations
OMIM 114610
References
Devane TIPS 15:40 1994