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bisacodyl (Dulcolax tablets, suppository)

Tradename: Dulcolax (tradename also used for other products). Indications: - relief of constipation - bowel preparation [4] Dosage: 1) 5-15 mg PO/PR BID PRN 2) 10 mg PO QD effective for constipation [3] Tabs: 5 mg. Suppositories: 10 mg. Pharmacokinetics: onset of bowel relief is 6-8 hours Mechanism of action: stimulant laxative

General

laxative

Properties

MISC-INFO: elimination route LIVER pregnancy-category + safety in lactation ?

Database Correlations

PUBCHEM correlations

References

  1. The Pharmacological Basis of Therapeutics, 9th ed. Gilman et al, eds. Permagon Press/McGraw Hill, 1996
  2. Drug Information & Medication Formulary, Veterans Affairs, Central California Health Care System, 1st ed., Ravnan et al eds, 1998
  3. Kamm MA et al. Oral bisacodyl is effective and well-tolerated in patients with chronic constipation. Clin Gastroenterol Hepatol 2011 Jul; 9:577. PMID: 21440672
  4. Deprecated Reference

Component-of

bisacodyl/c kit protein bisacodyl/citrate/magnesium carbonate/potassium citrate bisacodyl/citrate/magnesium carbonate/potassium citrate/suppository bisacodyl/polyethylene glycol/potassium chloride/sodium bicarbonate/sodium chloride bisacodyl/suppository