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adrenergic receptor
Related
Na+ dependent noradrenaline transporter; norepinephrine transporter; NET; solute carrier family 6 member 2 (SLC6A2, NAT1, NET1, SLC6A5)
norepinephrine; noradrenaline (Levophed)
Specific
alpha adrenergic receptor
beta adrenergic receptor
dopamine receptor
General
G-protein coupled receptor; serpentine receptor
Properties
COMPARTMENT: cellular membrane
MOTIF: exoplasmic domain {N-TERMINAL}
ligand-binding site
SITE: WITHIN-MEMBRANE-DOMAINS
FOR-BINDING-OF: norepinephrine
epinephrine
transmembrane domain {TM1}
transmembrane domain {TM2}
transmembrane domain {TM3}
transmembrane domain {TM4}
transmembrane domain {TM5}
transmembrane domain {TM6}
transmembrane domain {TM7}
transmembrane domain (7)
guanine nucleotide exchange domain
NAME: guanine nucleotide exchange domain
binding site
SITE: C-TERMINAL-CYS
EFFECTOR-BOUND: palmitate
BOUND-VIA: carboxylate
cytoplasmic domain {C-TERMINAL}
References
Weiss et al FASEB J 2:2841 1988