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adenosine diphosphate [ADP] receptor


Interactions

molecular events

Related

adenosine 5'-diphosphate (ADP)

Specific

P2Y12 purinoceptor; P2Y purinoceptor 12; P2Y12; P2Y12 platelet ADP receptor; P2Y(ADP); ADP-glucose receptor; ADP receptor P2Y12; ADPG-R; P2Y(AC); P2Y(cyc); P2T(AC); SP1999 (P2RY12, HORK3)

General

G-protein coupled receptor; serpentine receptor

Properties

COMPARTMENT: plasma membrane CELL: monocyte MOTIF: exoplasmic domain {N-TERMINAL} ligand-binding site transmembrane domain {TM1} transmembrane domain {TM2} transmembrane domain {TM3} transmembrane domain {TM4} transmembrane domain {TM5} transmembrane domain {TM6} transmembrane domain {TM7} transmembrane domain (7) guanine nucleotide exchange domain NAME: guanine nucleotide exchange domain binding site SITE: C-TERMINAL-CYS EFFECTOR-BOUND: palmitate BOUND-VIA: carboxylate cytoplasmic domain {C-TERMINAL}

References

- Altieri DC, Wiltse WL, Edgington TS. Signal transduction initiated by extracellular nucleotides regulates the high affinity ligand recognition of the adhesive receptor CD11b/CD18. J Immunol. 1990 Jul 15;145(2):662-70. PMID: 1973186